Liste des Publications[ McCurdy Christopher R.]

N,Ndimethylformamide.diiodine complex (DMF.I2) as an innovative efficient green catalyst in the synthesis of thiosemicarbazones by condensation of ketones with thiosemicarbazides

Kasséhin Urbain C. [1], Gbaguidi Fernand A. [2], McCurdy Christopher R. [3], Poupaert Jacques H. [4],

In a drug discovery program aimed at finding new anti-trypanosomal drugs, we developed the N, Ndimethylformamide.diiodine complex (DMF.I2) as an innov [...]

Article, Ajoutée le 17/01/2017 10:11

Insight into the Diels-Alder reaction: A green chemistry revisitation of the synthesis of a cantharidine-like trypanocidal pilot-molecule

Gbaguidi A. Fernand [1], Kasséhin Urbain C. [2], Prevost Julien R. C. [3], Frederick Raphaël [4], McCurdy Christopher R. [5], Poupaert Jacques H. [6],

Relying on a straightforward « Green-Chemistry » based approach, this article reports an optimized Diels-Alder (DA) experimental set-up allowing for t [...]

Article, Ajoutée le 17/01/2017 10:25

A concise synthesis of 2-(1,2,3,4-tetrahydro-6-methoxynaphthalen-4-yl) ethanamine, a key intermediate in the elaboration compound library of agomelatine analogs

Kasséhin Urbain C. [1], Gbaguidi A. Fernand [2], McCurdy Christopher R. [3], Poupaert Jacques H. [4],

Agomelatine, a melatonin-like antidepressant drug based on a naphthalene scaffold, has received considerable attention these last twenty years. This d [...]

Article, Ajoutée le 17/01/2017 10:32

Trypanocidal activity of a thioacyl-thiosemicarbazide derivative associating both immunostimulating thalidomide and anti-parasitic thiosemicarbazide pharmacophores

Kasséhin Urbain C. [1], Gbaguidi A. Fernand [2], McCurdy Christopher R. [3], Poupaert Jacques H. [4],

African trypanosomiasis remains a life-threatening disease and there is nowadays an urgent need for improved therapeutic agents for this pathology. In [...]

Article, Ajoutée le 17/01/2017 10:54

Synthesis of antitrypanosomal thiosemicarbazones using anthranilic acid as an innovative Green nucleophilic catalyst

Kasséhin Urbain C. [1], Gbaguidi A. Fernand [2], McCurdy Christopher R. [3], Poupaert Jacques H. [4],

Trypanosomiasis constitutes a severe health problem for sub-saharian African and latin American population and there is an urgent need for better drug [...]

Article, Ajoutée le 17/01/2017 11:37

Synthesis and Antiepileptic Activity Assessment of 5-Benzoyloxindole, a Novel Phenytoinergic Template

Kasséhin Urbain C. [1], Gbaguidi A. Fernand [2], Carato Pascal [3], McCurdy Christopher R. [4], Poupaert Jacques H. [5],

Based on a rational approach using merely bioisosterism as euristic tool, we designed and tested a short series of congeners of 6-benzoyl-2(3H)-benzox [...]

Article, Ajoutée le 18/01/2017 09:01

Electronic and steric effects in the control of the Anilinium chloride catalyzed condensation reaction between Aldones and 4-Phenylthiosemicarbazide

Kasséhin Urbain C. [1], Gbaguidi A. Fernand [2], Kapanda Coco N. [3], McCurdy Christopher R. [4], Bigot André K. [5], Poupaert Jacques H. [6],

A concise series of aldehydes and ketones were reacted in a condensation reaction with 4phenylthiosemicarbazide in order to assess the relative influe [...]

Article, Ajoutée le 18/01/2017 10:44

Is cocaine a social drug? Exploration of the stereo-structure of cocaine’s pharmacophore

Poupaert Jacques H. [1], Gbaguidi A. Fernand [2], Kapanda Coco N. [3], Aichaoui Hocine [4], McCurdy Christopher R. [5],

Based on a line of evidence (logP, pKa, 1H-, and 13C-NMR, and molecular modeling studies), it appears that cocaine undergoes a hydrophobic collapse wh [...]

Article, Ajoutée le 19/01/2017 10:29

Solid-Liquid Phase Transfer Catalysis and Microwave-Assisted Green Synthesis of Tetracyclone

Kasséhin Urbain C. [1], Gbaguidi A. Fernand [2], Carato Pascal [3], McCurdy Christopher R. [4], Accrombessi Georges C. [5], Poupaert Jacques H. [6],

A green synthesis of tetracyclone (2, 3, 4, 5-tetraphenyl-2, 4-cyclopentadien-1-one) has been conceived and executed on the basis of a rationale desig [...]

Article, Ajoutée le 25/01/2017 08:29

Publications par entité

  • Centre de Formation et de Recherche en matière de Population (CEFORP) (15)
  • Centre Interfacultaire de Formation et de Recherche en Environnement pour le Développement Durable (CIFRED) (18)
  • Chaire Internationale en Physique Mathématique et Applications (CIPMA-Chaire UNESCO) (16)
  • Ecole Nationale d'Administration et de Magistrature (ENAM) (47)
  • Ecole Nationle d'Economie Appliquée et de Management (81)
  • Ecole Normale Supérieure (24)
  • Ecole Polytechnique d'Abomey-Calavi (EPAC) (877)
  • Faculté de droit et de Science Politique (FADESP) (57)
  • Faculté des Lettres et Sciences Humaines (FLASH) (889)
  • Faculté des Sciences Agronomiques (1429)
  • Faculté des Sciences de la Santé (FSS) (1743)
  • Faculté des Sciences Economiques et de Gestion (FASEG) (143)
  • Faculté des Sciences et Techniques (FAST) (787)
  • Faculté des Sciences Humaines et Sociales (FASHS) (19)
  • Institut de Formation et de Recherche en Informatique (IFRI) (72)
  • Institut de Mathématiques et de Sciences Physiques (IMSP) (72)
  • Institut National de l'Eau (INE) (13)
  • Institut National des Métiers d'Art d'Archéologie et de la Culture (INMAAC) (4)
  • Institut National Médico Sanitaire ( INMeS) (0)
  • Institut Régional de Santé Publique (IRSP) (51)

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